Hexarelinwani roba nepeptide na sirri na hormone girma (GHS)kuma mai ikoBayani: GHSR-1A, ci gaba don tada hankalisakin hormone girma na endogenous (GH).. Nasa neghrelin mimetic iyalikuma ya ƙunshi amino acid guda shida (hexapeptide), yana ba da ingantaccen kwanciyar hankali na rayuwa da ƙarin tasirin sakin GH idan aka kwatanta da analogs na baya kamar GHRP-6.
Ana nazarin Hexarelin sosai don aikace-aikacen sa a cikiEndocrinology, zubar da tsoka, gyaran zuciya, da maganin tsufa, saboda ikonta na haɓaka GH da dabi'aInsulin-kamar girma factor 1 (IGF-1)matakan ba tare da gabatar da hormones na waje kai tsaye ba.
Hexarelin yana ɗaure zuwa gaMai karɓar mai karɓa na sirri na hormone girma (GHSR-1a)a kan pituitary da hypothalamus, mimicking mataki naghrelin- yunwar dabi'ar jiki da GH-sakin hormone.
Mahimman ayyukan physiological:
Yana ƙarfafa sakin GH mai bugun jini
Yana ƙara yawoFarashin IGF-1matakan
Yana haɓakaanabolic effects(girman tsoka, farfadowa)
Yana goyan bayanmai metabolismkumasabuntawar salula
Zai iya nunawacardioprotectivekumaanti-apoptotictasiri
Ba kamar sauran GHS peptides ba, Hexarelin yayiBa a ƙara yawan cortisol ko prolactin ba, yana ba da ingantaccen bayanin martabar endocrin.
Yana haɓakam jiki taroci gaba
Yana haɓakawagyaran tsoka da farfadowa
Ya yi karatu asarcopenia, cachexia, da farfadowa bayan tiyata
Nazarin preclinical ya nunaingantaccen aikin zuciyabayan myocardial rauni
Yana ragewacardiac fibrosisda haɓakawaɓangarorin fitar da huhu na hagu
Yiwuwar amfani a cikiciwon zuciyakumatsufa na zuciyasamfura
Yana ƙaruwalipolysiskuma yana ingantainsulin sensitivity
Yana goyan bayanmaganin tsufata hanyar GH / IGF-1 axis ƙarfafawa
Zai iya taimakawa kiyayewayawan kashi da lafiyar haɗin gwiwa
Tsafta ≥ 99%
An samar ta hanyarTsarin peptide mai ƙarfi (SPPS)
Matsayin GMP, ƙananan endotoxin da sauran sauran ƙarfi
Samfura mai sassauƙa:R&D zuwa sikelin kasuwanci