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Hexarelin

Takaitaccen Bayani:

Hexarelin shine peptide peptide hormone girma na roba (GHS) da kuma GHSR-1a agonist mai ƙarfi, wanda aka haɓaka don haɓaka haɓakar haɓakar hormone (GH). Yana cikin dangin ghrelin mimetic kuma ya ƙunshi amino acid shida (wani hexapeptide), yana ba da ingantaccen kwanciyar hankali na rayuwa da ƙarin tasirin sakin GH idan aka kwatanta da analogs na baya kamar GHRP-6.

Abubuwan API:

Tsafta ≥ 99%

Ana samarwa ta hanyar haɗakar peptide mai ƙarfi (SPPS)

Matsayi kamar GMP, ƙarancin endotoxin da ragowar sauran ƙarfi

Samfura mai sassauƙa: R&D zuwa sikelin kasuwanci


Cikakken Bayani

Tags samfurin

Hexarelin API - Bayanin Samfura

Hexarelinwani roba nepeptide na sirri na hormone girma (GHS)kuma mai ikoBayani: GHSR-1A, ci gaba don tada hankalisakin hormone girma na endogenous (GH).. Nasa neghrelin mimetic iyalikuma ya ƙunshi amino acid guda shida (hexapeptide), yana ba da ingantaccen kwanciyar hankali na rayuwa da ƙarin tasirin sakin GH idan aka kwatanta da analogs na baya kamar GHRP-6.

Ana nazarin Hexarelin sosai don aikace-aikacen sa a cikiEndocrinology, zubar da tsoka, gyaran zuciya, da maganin tsufa, saboda ikonta na haɓaka GH da dabi'aInsulin-kamar girma factor 1 (IGF-1)matakan ba tare da gabatar da hormones na waje kai tsaye ba.


Tsarin Aiki

Hexarelin yana ɗaure zuwa gaMai karɓar mai karɓa na sirri na hormone girma (GHSR-1a)a kan pituitary da hypothalamus, mimicking mataki naghrelin- yunwar dabi'ar jiki da GH-sakin hormone.

Mahimman ayyukan physiological:

  • Yana ƙarfafa sakin GH mai bugun jini

  • Yana ƙara yawoFarashin IGF-1matakan

  • Yana haɓakaanabolic effects(girman tsoka, farfadowa)

  • Yana goyan bayanmai metabolismkumasabuntawar salula

  • Zai iya nunawacardioprotectivekumaanti-apoptotictasiri

Ba kamar sauran GHS peptides ba, Hexarelin yayiBa a ƙara yawan cortisol ko prolactin ba, yana ba da ingantaccen bayanin martabar endocrin.


Bincike da Yiwuwar Jiyya

1. Girman tsoka & Farfadowa

  • Yana haɓakam jiki taroci gaba

  • Yana haɓakawagyaran tsoka da farfadowa

  • Ya yi karatu asarcopenia, cachexia, da farfadowa bayan tiyata

2. Kariya na zuciya

  • Nazarin preclinical ya nunaingantaccen aikin zuciyabayan myocardial rauni

  • Yana ragewacardiac fibrosisda haɓakawaɓangarorin fitar da huhu na hagu

  • Yiwuwar amfani a cikiciwon zuciyakumatsufa na zuciyasamfura

3. Fat Metabolism & Anti-tsufa

  • Yana ƙaruwalipolysiskuma yana ingantainsulin sensitivity

  • Yana goyan bayanmaganin tsufata hanyar GH / IGF-1 axis ƙarfafawa

  • Zai iya taimakawa kiyayewayawan kashi da lafiyar haɗin gwiwa


Siffofin API (Rukunin Gentolex)

  • Tsafta ≥ 99%

  • An samar ta hanyarTsarin peptide mai ƙarfi (SPPS)

  • Matsayin GMP, ƙananan endotoxin da sauran sauran ƙarfi

  • Samfura mai sassauƙa:R&D zuwa sikelin kasuwanci


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