Melanotan IIshine analog na heptapeptide synthetic cyclicα-melanocyte-stimulating hormone (α-MSH), ci gaba zuwainganta melanogenesis, ingantaKariyar UV, da daidaitawaayyukan jima'i da na rayuwa. Yana aiki azaman aagonist mara zabina masu karɓar melanocortin, musammanSaukewa: MC1R, Saukewa: MC3R, kumaSaukewa: MC4R.
Asali ya yi karatu domin satanningkumaphotoprotectiveProperties, Melanotan II ya kuma nuna tasiri a kaninganta libido, rage cin abinci, kumamakamashi balance, Yin shi peptide bincike na multifunctional tare da sha'awar dermatology, endocrinology, da magungunan jima'i.
Melanotan II yana aiki ta hanyar kunna masu karɓar melanocortin da yawa:
Saukewa: MC1R: Yana kara kuzarisamar da melanin→ yana ƙara launin fata da kariya ta UV
Saukewa: MC3R/MC4R: Shiga cikikula da ci, inganta libido, kumamakamashi homeostasis
Ketare shingen kwakwalwar jini, rinjayar tsakiyar neurohormonal hanyoyin
Kodayake ba a yarda da amfani da magani ba, Melanotan II ana nazarin ko'ina don masu zuwa:
Yana haɓakaeumelanin kira, kai gatanning na halitta
Yana bayarwatasirin kariya na hotoba tare da fallasa rana ba
Mai yuwuwa don rage haɗarin kansar fata a cikin mutane masu fata
An nuna wayana kara sha'awa da sha'awar jima'ia cikin maza da mata
Ya yi karatu a matsayin mai yuwuwar magani gaRashin karfin mazakuta (ED)ta MC4R kunnawa
Mayurage ci da abincita hanyar yin aiki akan hanyoyin hypothalamic
Mai yuwuwar haɗin gwiwa a cikibinciken kiba
Babban tsarki ≥ 99%(HPLC & LC-MS sun tabbatar)
Haɗa ta hanyarTsarin peptide mai ƙarfi (SPPS)
Low endotoxin, ƙananan sauran kaushi
Akwai a cikiR&D zuwa sikelin kasuwanci