Suna | Pregabalin |
Lambar CAS | 148553-8-8 |
Tsarin kwayoyin halitta | C8h17No2 |
Nauyi na kwayoyin | 159.23 |
Lambar Einecs | 604-639-1 |
Tafasa | 274.0 ± 23.0 ° C |
M | 98% |
Ajiya | Rufe a bushe, zazzabi dakin |
Fom | Foda |
Launi | Farin launi |
Shiryawa | Jag Bag + Aluminum Jakar |
3 (s) - (Aminomethyl) -5-methylhexanoic acid; (3s) -3-3- (aminomathyl) -5-methyhyl) -5-methyhyl) -5-methylin-hexanoic ) -Pregabalin; (s) -pregabal
Tasirin magunguna
Pregabalin yana da kyakkyawan tasirin warkewa a kan popilesy. Bincike akan nau'ikan cututtukan dabbobi daban-daban sun nuna cewa progabalin zai iya hana epilptic seizures, da kashi na aiki shine 3-10 sau da yawa fiye da na gepentin. Nazarin sun gano cewa progabalin zai iya rage azzalumi da kuma motsin igiyar igiyar ruwa na bera da ciwon sukari, da kuma hana zafin da ya shafi lalacewa kashin baya. Halin. Nazarin dabbobi sun gano cewa progabalin na iya samun fa'idodi a hade tare da opiiids. Pregabalin yana ba da sabon zaɓi don maganin asibiti na cututtukan zafi.
Inji
Pregabalin na iya rage sakin alli na wasu 'yan jihar Neurotransmited ta modulating aikin tashar. Ko da yake Pregabalin yana da matuƙar yin ta'addanci na inhihibransmiter γ-aminobutyric γ-aminobutyric γ-amar), baya ƙara haɗuwa a cikin al'adun garga a cikin Kwastam na berayen, kuma ba shi da mummunan tasiri a Gaba Uptake ko lalata. Koyaya, binciken ya gano cewa tsawan tsawan lokaci na al'adun gargajiya don pregabalin ya ƙara yawan jigilar hanyoyin tallafi na Giba da kuma ragin jigilar kayayyaki na Giba. Pregabalin ba ya toshe tashoshin sodium, ba shi da wani aiki a kan masu karɓar Opoloid, baya canza ayyukan ta dopamine, herotonin, ko norepinephrine. Shiga.
Kwarewar magani
1. Ba a haɗa shi ta tsarin Cytochrromer P450 na Cytolen, saboda haka, da wuya ya yi hulɗa tare da wasu magunguna. Ba ya shafar ƙwayar magunguna na magunguna masu maganin cututtukan magunguna (kamar ƙwayoyin ƙwayar ƙwayar sodium, Phennoin, Carbaazepine, wakilai na baki, diuretics, da insulin.
2. Lokacin da ake amfani da wannan samfurin tare da oxycodone, aikin sanannen aikin za a rage da lalacewa ta aikin motsi da kuma za a inganta lalacewa.
3. Yana da tasiri sosai tare da lorazepam da ethanol.