Kayayyaki
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Saukewa: CJC-1295
An samar da CJC-1295 API ta amfani da fasaha mai ƙarfi peptide synthesis (SPPS) kuma an tsarkake ta ta amfani da HPLC don cimma babban tsafta da daidaiton tsari-zuwa-tsari.
Siffofin samfur:Tsafta ≥ 99%
Low ragowar kaushi da nauyi karafa
Endotoxin-free, mara-immunogenic hanyar kira
Abubuwan da za a iya daidaita su: mg zuwa kg
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NAD+
Abubuwan API:
Babban tsarki ≥99%
Pharmaceutical-grade NAD+
Matsayin masana'anta kamar GMP
NAD+ API yana da kyau don amfani a cikin abubuwan gina jiki, alluran allura, da manyan hanyoyin kwantar da hankali na rayuwa.
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Boc-Tyr(tBu)-Aib-Glu(OtBu) -Gly-OH
Boc-Tyr(tBu)-Aib-Glu(OtBu) -Gly-OHwani tetrapeptide ne mai kariya wanda aka saba amfani dashi a cikin binciken haɗin peptide. Ƙungiyoyin Boc (tert-butyloxycarbonyl) da tBu (tert-butyl) suna zama ƙungiyoyi masu kariya don hana halayen gefe yayin taron sarkar peptide. Haɗin Aib (α-aminoisobutyric acid) yana taimakawa wajen haifar da sifofin helical da haɓaka kwanciyar hankali na peptide. Ana nazarin wannan jeri na peptide don yuwuwar sa a cikin bincike mai daidaituwa, nadewa peptide, da kuma matsayin tubalin gini don haɓaka peptides na bioactive tare da ingantaccen kwanciyar hankali da ƙayyadaddun bayanai.
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Cagrilintide
Cagrilintide wani agonist na amylin mai karɓa ne na roba, mai ɗaukar lokaci mai tsawo wanda aka haɓaka don kula da kiba da rikice-rikice masu alaƙa da nauyi. Ta hanyar kwaikwayon amylin hormone na halitta, yana taimakawa wajen daidaita sha'awa, jinkirin zubar da ciki, da haɓaka jin dadi. Babban tsaftar Cagrilintide API ɗinmu an samar da shi ta hanyar haɗin sinadarai kuma ya dace da ma'aunin ƙimar magunguna, yana mai da shi dacewa don amfani a cikin ƙirar sarrafa nauyi na ci gaba.
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Tesamorelin
Tesamorelin API yana amfani da fasaha mai ƙarfi mai ƙarfi peptide synthesis (SPPS) kuma yana da fasali masu zuwa:
Tsafta ≥99% (HPLC)
Babu endotoxin, karafa masu nauyi, sauran kaushi da aka gwada
Amino acid jerin da tsarin da LC-MS/NMR ya tabbatar
Samar da keɓaɓɓen samarwa a cikin gram zuwa kilogiram -
Fmoc-Ile-Aib-OH
Fmoc-Ile-Aib-OH tubalin ginin dipeptide ne da ake amfani da shi a cikin haɗakar peptide mai ƙarfi (SPPS). Ya haɗu da isoleucine mai kariya na Fmoc tare da Aib (α-aminoisobutyric acid), amino acid wanda ba na halitta ba wanda ke haɓaka kwanciyar hankali na helix da juriya na protease.
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Fmoc-L-Lys[Eic(OtBu)-γ-Glu(OtBu)-AEEA-AEEA]-OH
Fmoc-L-Lys [Eic(OtBu)-γ-Glu(OtBu) -AEEA-AEEA] -OH tubalin ginin amino acid ne mai aiki wanda aka ƙera don isar da magunguna da aka yi niyya da haɓakar halittu. Yana fasalta nau'in Eic (eicosanoid) don hulɗar lipid, γ-Glu don niyya, da AEEA sarari don sassauci.
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Boc-Tyr (tBu) - Aib-OH
Boc-Tyr (tBu) -Aib-OH wani shingen ginin dipeptide mai kariya wanda aka yi amfani dashi a cikin haɗin peptide, yana haɗa Boc-protected tyrosine da Aib (α-aminoisobutyric acid). Ragowar Aib yana haɓaka samuwar helix da juriya na protease.
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Boc-His(Trt)-Ala-Glu(OtBu)-Gly-OH
Boc-His (Trt) -Ala-Glu (OtBu) - Gly-OH wani yanki ne mai kariya na tetrapeptide wanda aka yi amfani da shi a cikin haɓakar peptide mai ƙarfi (SPPS) da ci gaban peptide miyagun ƙwayoyi. Ya haɗa da ƙungiyoyin karewa don haɗakarwa ta orthogonal kuma yana fasalta jeri mai amfani a ƙirar bioactive da tsarin peptide.
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Fmoc-Lys(Pal-Glu-OtBu) -OH
Fmoc-Lys(Pal-Glu-OtBu) -OH ƙwararren ginin amino acid ne na lipid wanda aka tsara don haɗuwa da peptide-lipid. Yana da fasalin lysine mai kariya ta Fmoc tare da sarkar gefen palmitoyl-glutamate, yana haɓaka alaƙar membrane da bioavailability.
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Fmoc-His-Aib-OH
Fmoc-His-Aib-OH shine toshe ginin dipeptide da aka yi amfani da shi a cikin kirar peptide, yana haɗa Fmoc-protected histidine da Aib (α-aminoisobutyric acid). Aib yana gabatar da rigidity mai daidaituwa, yana mai da shi mahimmanci don ƙirƙira helical da tsayayyen peptides.
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Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH
Boc-His (Trt) -Aib-Glu (OtBu) - Gly-OH wani yanki ne na tetrapeptide mai kariya wanda aka yi amfani dashi a cikin haɗin peptide da ci gaban ƙwayoyi. Ya ƙunshi ƙungiyoyin ayyuka masu kariya da dabaru don haɗin kai na mataki-mataki da fasali Aib (α-aminoisobutyric acid) don haɓaka kwanciyar hankali na helix da rigidity mai daidaitawa.
