| Suna | Farashin RU-58841 |
| Lambar CAS | 154992-24-2 |
| Tsarin kwayoyin halitta | Saukewa: C17H18F3N3O3 |
| Nauyin kwayoyin halitta | 369.34 |
| Lambar EINECS | 1592732-453-0 |
| Wurin Tafasa | 493.6± 55.0 °C (An annabta) |
| Yawan yawa | 1.39 |
| Yanayin ajiya | An rufe shi a bushe, adana a cikin injin daskarewa, ƙasa da -20 ° C |
| Siffar | Foda |
| Launi | Fari |
| Shiryawa | PE bag+Aluminum bag |
RU58841. onitrile; 4- [3- (4-Hydroxybutyl) -4,4-diMethyl-2,5-dioxoiMidazolidin-1-yl]-2- (trifluoroMethyl) ben zonitrile; RU-58841E: candyli (at) speedgainpharma (dot) com; CS-637; RU588841; RU58841; RU58841; RU-58841
Bayani
RU 58841 (PSK-3841) antagonist mai karɓar mai karɓar androgen ne wanda ke haɓaka haɓakar gashi.RU58841 magani ne na bincike da aka kirkira don maganin alopecia na androgenic, wanda kuma aka sani da gashin gashi na maza (MPD).
A matsayin maganin anti-androgen na gaba, ka'idodin aikinsa ba daidai ba ne da na finasteride. Finasteride kai tsaye yana aiki akan 5a reductase, yana hana canjin testosterone zuwa DHT, kuma yana rage abun ciki na DHT a cikin jiki. RU58841 yana toshe hulɗar tsakanin dihydrotestosterone da masu karɓar gashin gashi, ba kai tsaye ya rage abun ciki na DHT ba, amma yana rage ɗaurin DHT da masu karɓar gashin gashi, don cimma manufar magance alopecia na androgenetic.
4-[3- (4-Hydroxybutyl) -4,4-dimethyl-2,5-dioxo-1-imidazolidinyl] -2- (trifluoromethyl) benzonitrile za a iya amfani dashi azaman magani Chemical kira tsaka-tsaki.Idan 4-[3- (4-hydroxybutyl) -4,4-dimethyl-2,5-dioxo-1-imidazolidinyl] -2- (trifluoromethyl) benzonitrile an shayar da shi, Matsar da mai haƙuri zuwa iska mai kyau;Idan an samu fata, a cire gurɓatattun tufafi, a wanke fata sosai da sabulu da ruwa, sannan a nemi kulawar likita idan rashin jin daɗi ya faru;
Tasirin Side
Ana shafa RU58841 a fatar kan mutum, a shayar da shi a cikin gashin kansa, kuma a ka'idar, yana iya shiga cikin jini kuma yana shafar wasu sassan jiki. Amma ba a sami sakamako mai illa ba a cikin nazarin aikace-aikacen da ake amfani da su a cikin birai. Duk da haka, wasu mutanen da suka gwada RU58841 suna da'awar cewa sun sami wasu sakamako masu illa daga amfani da RU, ciki har da fushin fata, rage yawan libido, rashin barci, tashin zuciya, jajayen idanu, dizziness, da ciwon kai.