• Shugaban_BANGER_01

Deflazackort yana da anti-mai kumburi, anti-rashin lafiyan ƙwayar cuta, da kuma ƙara yawan tasirin gluconeogenis

A takaice bayanin:

Maɗaukaki: 255-256.5 ° C

Takamaiman juyawa: d + 62.3 ° (c = 0 5chloroform)

Bhafi na: 595.4 ± 50.0 ° C (annabta)

Density: 1.41

Yanayin ajiya: 2-8 ° C

Sulquility: DMSO: ≥20mg / ml

Maɗaukaki mai tsabta: (Pka) 14.30 ± 0.70 (annabta)

Form: foda

Launi: Baki


Cikakken Bayani

Tags samfurin

Cikakken Bayani

Suna Deflazackort
Lambar CAS 14484-4-0-0
Tsarin kwayoyin halitta C25H31NO6
Nauyi na kwayoyin 441.52
Lambar Einecs 238-483-7
Tafasa 595.4 ± 50.0 ° C
M 98%
Ajiya Rufe a bushe, zazzabi dakin
Fom Foda
Launi Farin launi
Shiryawa Jag Bag + Aluminum Jakar

Kwatanci

16-d) oxazole-3,20 11F-hydroxy-21-Acetyloxy-21-metyl-1,2,4,5-Titrordhydrogroveno [17,2,4,5-DORTHole-3,20-Dione; (5'β) -21-hydroxy -# Methylpregnano [17,16-D] oxazole-1,4-Dione-3,20-Dione; 11b, 21-Dihydroxy-2 '-; Denazackort

Tasirin magunguna

Alamar
Don firam na farko ko sakandare Adrenal isa na biyu, rheumatism, cututtukan ƙwayar cuta, cututtukan ƙwayar cuta, cututtukan cututtukan jini, da kuma haɗin cutar cututtukan ƙwayar cuta, da kuma haɗin cutar cututtukan ƙwayar cuta, da kuma a cikin cututtukan ƙwayar cuta, da kuma haɗawa da cututtukan ƙwayar cuta da kuma rarraba cututtukan ƙwayar cuta.

Matakan kariya
(1) Kamar sauran glucocorticoids, yana contraindicated ga cututtukan cututtukan cututtuka.
(2) Yi amfani da taka tsantsan a cikin tiyata na rarrabuwa, gazawar Gastrointestalin, gazawar koda, ciwon sukari, ciwon sukari, ciwon sukari, cututtukan osteoporosis, masu ciwon sukari da sauran cututtuka. Mata masu juna biyu da kuma lactating amfani da taka tsantsan.

Kwarewar magani
1. Deflazackort yana da tasirin fitowar potassium, don haka ya kamata a ɗauki kulawa lokacin da ake amfani da shi a haɗe tare da diuretics.
2. Lokacin da aka yi amfani da shi a hade tare da kwayoyi tare da aikin enzymatic (Ribampin, Phenobarbital, da sauransu), ya kamata a ƙara gluctocorticoid da ta dace.
3. Erythromycin da Estrogen na iya hana metabolism na wannan samfurin da abubuwa masu aiki, kuma ya kamata a rage yawan abubuwa lokacin da aka yi amfani da shi. Kayan sunadarai Acetone-Hexane Crystallization, Melting Point 255-256.5 ℃. [α] d + 62.3 ° (c = 0.5, chloriform).

Amfani
Gluctocorts na zamani na uku na zamani suna da anti-mai kumburi, anti-rashin lafiyan ƙwayar cuta, da kuma ƙara yawan tasirin gluconeogenis. Don firamare da sakandare na sakandare, rheumatism, cututtukan fata, cuta, cuta ta cututtukan fata, da colitiscastic nephrotic syndromes, cututtukan mahaifa, da sauransu.


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