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Pharma APIs

  • Fmoc-His-Aib-OH

    Fmoc-His-Aib-OH

    Fmoc-His-Aib-OH shine toshe ginin dipeptide da aka yi amfani da shi a cikin kirar peptide, yana haɗa Fmoc-protected histidine da Aib (α-aminoisobutyric acid). Aib yana gabatar da rigidity mai daidaituwa, yana mai da shi mahimmanci don ƙirƙira helical da tsayayyen peptides.

  • Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH

    Boc-His(Trt)-Aib-Glu(OtBu)-Gly-OH

    Boc-His (Trt) -Aib-Glu (OtBu) - Gly-OH wani yanki ne na tetrapeptide mai kariya wanda aka yi amfani dashi a cikin haɗin peptide da ci gaban ƙwayoyi. Ya ƙunshi ƙungiyoyin ayyuka masu kariya da dabaru don haɗin kai na mataki-mataki da fasali Aib (α-aminoisobutyric acid) don haɓaka kwanciyar hankali na helix da rigidity mai daidaitawa.

  • Ste-γ-Glu-AEEA-AEEA-OSU

    Ste-γ-Glu-AEEA-AEEA-OSU

    Ste-γ-Glu-AEEA-AEEA-OSU sinadari ne na roba mai haɗaɗɗiyar ƙwayar cuta wanda aka ƙera don isar da magunguna da aka yi niyya da haɗin gwiwar magungunan-magungunan (ADCs). Yana fasalta wutsiya ta stearoyl (Ste) hydrophobic, γ-glutamyl manufa motif, AEEA spacers don sassauci, da ƙungiyar OSu (NHS ester) don ingantaccen haɗin gwiwa.

  • Fmoc-Ile-αMeLeu-Leu-OH

    Fmoc-Ile-αMeLeu-Leu-OH

    Fmoc-Ile-αMeLeu-Leu-OH wani shingen gini ne na roba mai kariya na tripeptide wanda ke nuna α-methylated leucine, wanda aka saba amfani dashi a ƙirar magungunan peptide don haɓaka kwanciyar hankali na rayuwa da zaɓin mai karɓa.

  • Dodecyl Phosphocholine (DPC)

    Dodecyl Phosphocholine (DPC)

    Dodecyl Phosphocholine (DPC) wani wanki ne na roba na roba wanda aka yi amfani dashi sosai a cikin binciken furotin na membrane da tsarin tsarin halitta, musamman a cikin NMR spectroscopy da crystallography.

  • Caspofungin don kamuwa da cututtukan fungal

    Caspofungin don kamuwa da cututtukan fungal

    Suna: Caspofungin

    Lambar CAS: 162808-62-0

    Tsarin kwayoyin halitta: C52H88N10O15

    Nauyin Kwayoyin: 1093.31

    Lambar EINECS: 1806241-263-5

    Matsayin tafasa: 1408.1 ± 65.0 °C (An annabta)

    Yawan yawa: 1.36± 0.1 g/cm3(an annabta)

    Adadin acidity: (pKa) 9.86± 0.26 (an annabta)

  • Daptomycin 103060-53-3 don Cututtuka masu Yaduwa

    Daptomycin 103060-53-3 don Cututtuka masu Yaduwa

    Suna: Daptomycin

    Lambar CAS: 103060-53-3

    Tsarin kwayoyin halitta: C72H101N17O26

    Nauyin Kwayoyin: 1620.67

    Lambar EINECS: 600-389-2

    Matsayin narkewa: 202-204 ° C

    Matsayin tafasa: 2078.2 ± 65.0 °C (An annabta)

    Yawan yawa: 1.45± 0.1 g/cm3(an annabta)

    Matsakaicin walƙiya: 87 ℃

  • Micafungin don antifungal da antiviral

    Micafungin don antifungal da antiviral

    Suna: Micafungin

    Lambar CAS: 235114-32-6

    Tsarin kwayoyin halitta: C56H71N9O23S

    Nauyin Kwayoyin: 1270.28

    Lambar EINECS: 1806241-263-5

  • Vancomycin shine maganin rigakafi na glycopeptide da ake amfani dashi don maganin rigakafi

    Vancomycin shine maganin rigakafi na glycopeptide da ake amfani dashi don maganin rigakafi

    Suna: Vancomycin

    Lambar CAS: 1404-90-6

    Tsarin kwayoyin halitta: C66H75Cl2N9O24

    Nauyin Kwayoyin: 1449.25

    Lambar EINECS: 215-772-6

    Maɗaukaki: 1.2882 (ƙididdigar ƙima)

    Fihirisar magana: 1.7350 (ƙididdiga)

    Yanayin ajiya: An rufe shi a bushe, 2-8 ° C

  • Vardenafil Dihydrochloride Maganin Rashin Matsala 224785-91-5

    Vardenafil Dihydrochloride Maganin Rashin Matsala 224785-91-5

    Lambar CAS: 224785-91-5

    Tsarin kwayoyin halitta: C23H32N6O4S

    Nauyin Kwayoyin: 488.6

    Lambar EINECS: 607-088-5

    Matsayin narkewa: 230-235 ° C

    Yawan yawa: 1.37

    Filashin wuta: 9 ℃

    Yanayin ajiya: An rufe shi a bushe, Ajiye a cikin injin daskarewa, ƙasa da -20 ° C

    Adadin acidity: (pKa) 9.86± 0.20 (an annabta)

  • Orlistat 96829-58-2 Rage Shayar da Fat ɗin Sietary, Sakamakon Rage Nauyi

    Orlistat 96829-58-2 Rage Shayar da Fat ɗin Sietary, Sakamakon Rage Nauyi

    Lambar CAS: 96829-58-2

    Tsarin kwayoyin halitta: C29H53NO5

    Nauyin Kwayoyin: 495.73

    Lambar EINECS: 639-755-1

    Takamaiman juyawa: D20-32.0°(c=1inchloroform)

    Matsayin tafasa: 615.9± 30.0°C (An annabta)

    Yawan yawa: 0.976± 0.06g/cm3(an annabta)

    Yanayin ajiya: 2-8°C

     

  • RU-58841 Anyi Amfani dashi azaman Rigakafin Asarar Gashi da Bakin Ƙirar Namiji

    RU-58841 Anyi Amfani dashi azaman Rigakafin Asarar Gashi da Bakin Ƙirar Namiji

    Lambar CBN: CB51396657

    Saukewa: RU58841

    Lambar CAS: 154992-24-2

    Tsarin kwayoyin halitta: C17H18F3N3O3

    Nauyin Kwayoyin: 369.34

    Lambar EINECS: 1592732-453-0