Suna | Sodium tianepine |
Lambar CAS | 66981-73-5-5 |
Tsarin kwayoyin halitta | C21H25CLN2O4S |
Nauyi na kwayoyin | 436.95200 |
Mallaka | 129-131 ° C |
Tafasa | 609.2ºC a 760 mmhg |
M | 99% |
Ajiya | Rufe a bushe, zazzabi dakin |
Fom | Foda |
Launi | Farin launi |
Shiryawa | Jag Bag + Aluminum Jakar |
Tianeptina; Tianetina [Inn-Spanish]; CoAxil; Tianeotine; Tianeotine; Tianeotine; Tianeotine; Tianeotine; Tianeotine; Tianeotine;
Amfani
Yana da yafi aiki akan tsarin 5-HT, ba tare da farin ciki ba, kwayar, Cedation, umetlcholine da cututtukan zuciya. Domin baƙin ciki.
Tasirin magunguna
1. Hanyar magangwama ta wannan samfurin ta bambanta da na Tca na gargajiya. Zai iya ƙara UPTake na 5-ht a cikin Synátiks Cleft, amma yana da sakamako mai rauni a kan Reuptake na 5-ht da na. Na iya haifar da tasirin haɓaka 5-ht neurinal watsawa. Ba shi da kusanci ga masu maye, H1, α1 da α2 - masu karɓar.
2. Ingancin wannan samfurin yayi kama da na tca, da amincinsa da irinsa sun fi tca (tricycressepressants). Ingancin wannan samfurin ya yi kama da na SSRIREXETINE.
3. Gwajin magunguna na dabbobi sun nuna cewa zai iya: Coarara ayyukan ƙwayoyin pyramidal a cikin hippocampus da hanzarta dawo da aikinta bayan hanawa; Theara yawan Reabsorption 5-hydroxytryptamine ta neurons a cikin cortex cardex da kuma hippocampus.
Karatun guba
- A hankali, gwaji na dogon lokaci: Babu canje-canje a cikin ilimin halitta, aikin hanta, ƙwararru na jini.
- Yin haifuwa na haihuwa da Taro: Tiannepine ba shi da tasiri a kan iyawar iyaye da aka bi da bi da kuma zuriyar da zuriya.
- Gwajin mutonajin: Tiannepine ba shi da tasirin mutonic.