• Shugaban_BANGER_01

Tianepine sodium don m aukuwa

A takaice bayanin:

Bayyanar da kaddarorin: farin m

Yankana: 1.38 g / cm3

Maɗaukaki: 129-131 ° C

Bhafi Point: 609.2ºC a 760 mmhg

Fasaha: 322.2ºC

Indextive Index: 1.639

Lambar CAS: 66981-73-5

Tsarin Abinci: C21H25Cl2o4S

Nauyi na kwayoyin: 436.95200


Cikakken Bayani

Tags samfurin

Cikakken Bayani

Suna Sodium tianepine
Lambar CAS 66981-73-5-5
Tsarin kwayoyin halitta C21H25CLN2O4S
Nauyi na kwayoyin 436.95200
Mallaka 129-131 ° C
Tafasa 609.2ºC a 760 mmhg
M 99%
Ajiya Rufe a bushe, zazzabi dakin
Fom Foda
Launi Farin launi
Shiryawa Jag Bag + Aluminum Jakar

Kwatanci

Tianeptina; Tianetina [Inn-Spanish]; CoAxil; Tianeotine; Tianeotine; Tianeotine; Tianeotine; Tianeotine; Tianeotine; Tianeotine;

Tasirin magunguna

Amfani

Yana da yafi aiki akan tsarin 5-HT, ba tare da farin ciki ba, kwayar, Cedation, umetlcholine da cututtukan zuciya. Domin baƙin ciki.

 

Tasirin magunguna

1. Hanyar magangwama ta wannan samfurin ta bambanta da na Tca na gargajiya. Zai iya ƙara UPTake na 5-ht a cikin Synátiks Cleft, amma yana da sakamako mai rauni a kan Reuptake na 5-ht da na. Na iya haifar da tasirin haɓaka 5-ht neurinal watsawa. Ba shi da kusanci ga masu maye, H1, α1 da α2 - masu karɓar.
2. Ingancin wannan samfurin yayi kama da na tca, da amincinsa da irinsa sun fi tca (tricycressepressants). Ingancin wannan samfurin ya yi kama da na SSRIREXETINE.
3. Gwajin magunguna na dabbobi sun nuna cewa zai iya: Coarara ayyukan ƙwayoyin pyramidal a cikin hippocampus da hanzarta dawo da aikinta bayan hanawa; Theara yawan Reabsorption 5-hydroxytryptamine ta neurons a cikin cortex cardex da kuma hippocampus.

 

Karatun guba

- A hankali, gwaji na dogon lokaci: Babu canje-canje a cikin ilimin halitta, aikin hanta, ƙwararru na jini.
- Yin haifuwa na haihuwa da Taro: Tiannepine ba shi da tasiri a kan iyawar iyaye da aka bi da bi da kuma zuriyar da zuriya.
- Gwajin mutonajin: Tiannepine ba shi da tasirin mutonic.


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